SCHEMBL28501237

SCHEMBL28501237

O=[N+]([O-])c1c(F)cccc1N1CCNCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.51
HTR7 P34969 5/20 0.51
LMNA P02545 1/20 0.51
GAA P10253 1/20 0.51
ALDH1A1 P00352 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ADRB1 P08588 4/20 0.46
SIRT6 Q8N6T7 1/20 0.46
HTR1A P08908 5/20 0.45
HTR3A P46098 2/20 0.45
HTR6 P50406 2/20 0.45
HTR2B P41595 1/20 0.45
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 1/20 0.44
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30480462 1.00 MAPT (0.51) MAPTHTR7LMNAGAAALDH1A1
Tert-Butyl Formate SCHEMBL27737428 0.87 MAPT (0.41) MAPTHTR7LMNAGAAALDH1A1
SCHEMBL23997432 0.86 MAPT (0.48) MAPTLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL30336949 0.86 MAPT (0.48) MAPTLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL3541135 0.84 MAPK1 (0.49) MAPTLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL8589619 0.83 ADRB1 (0.61) HTR7ALDH1A1ADRB1SIRT6HTR1A
SCHEMBL6663091 0.83 MAPT (0.52) MAPTHTR7LMNAGAAALDH1A1
SCHEMBL7374611 0.82 HTR7 (0.51) MAPTHTR7LMNAGAAALDH1A1
SCHEMBL9059492 0.82 ALDH1A1 (0.52) MAPTLMNAGAAALDH1A1CYP1A2
SCHEMBL31321242 0.78 ALDH1A1 (0.43) MAPTLMNAGAAALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112041300-B Indole and benzimidazole derivatives as dual 5-HT2A and 5-HT6 receptor antagonists 阿达梅德制药公司 2023-07-28 CN disclosed
CN-112041300-A Indole and benzimidazole derivatives as dual 5-HT2A and5-HT 6receptor antagonists 阿达梅德制药公司 2020-12-04 CN disclosed