SCHEMBL28501723

SCHEMBL28501723

CN1C(=O)c2cc(Br)cc3c([N+](=O)[O-])ccc1c23

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 2/20 0.43
CASP1 P29466 1/20 0.43
CASP3 P42574 1/20 0.43
CASP4 P49662 1/20 0.43
CASP7 P55210 1/20 0.43
CASP9 P55211 1/20 0.43
GAA P10253 2/20 0.41
NR1H2 P55055 2/20 0.40
NR1H3 Q13133 2/20 0.40
ACHE P22303 1/20 0.39
S100A4 P26447 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
MEN1 O00255 5/20 0.38
KMT2A Q03164 5/20 0.38
RAB9A P51151 3/20 0.38
NPC1 O15118 2/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
LMNA P02545 3/20 0.36
POLB P06746 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9290406 0.79 MEN1 (0.61) CASP6GAAMEN1KMT2ARAB9A
SCHEMBL28500614 0.74 MAPT (0.38) CASP6CASP1CASP3CASP4CASP7
SCHEMBL28490501 0.72 GABRA1 (0.42) CASP3ACHES100A4TRPV1MEN1
SCHEMBL7703726 0.70 S100A4 (0.44) GAAACHES100A4TRPV1MEN1
SCHEMBL7709778 0.69 ALDH1A1 (0.45) GAAACHES100A4TRPV1MEN1
SCHEMBL7706804 0.68 HTT (0.47) CASP6GAAACHEMEN1KMT2A
SCHEMBL7484059 0.68 MEN1 (0.61) CASP6GAAMEN1KMT2ARAB9A
SCHEMBL8618712 0.67 MEN1 (0.73) GAAMEN1KMT2ARAB9ANPC1
SCHEMBL20033849 0.66 MEN1 (0.41) CASP6CASP1CASP3CASP4CASP7
SCHEMBL7485990 0.65 MEN1 (0.61) CASP6GAAMEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112125885-A Benzoindole bifunctional molecular derivative and preparation method and application thereof 中国药科大学 2020-12-25 CN disclosed