SCHEMBL7709778

SCHEMBL7709778

C=CCON1C(=O)c2ccc([N+](=O)[O-])c3cc(Br)cc(c23)C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
MEN1 O00255 11/20 0.40
KMT2A Q03164 11/20 0.40
NPC1 O15118 6/20 0.40
RAB9A P51151 4/20 0.40
HTT P42858 5/20 0.38
ACHE P22303 1/20 0.36
POLB P06746 7/20 0.36
NPSR1 Q6W5P4 5/20 0.36
CCR6 P51684 3/20 0.36
LMNA P02545 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
PABPC1 P11940 2/20 0.36
TLR9 Q9NR96 2/20 0.36
S100A4 P26447 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
S1PR4 O95977 3/20 0.35
S1PR1 P21453 3/20 0.35
HPGD P15428 1/20 0.35
XBP1 P17861 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7706707 0.87 ALDH1A1 (0.45) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL7706804 0.81 HTT (0.47) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL7709710 0.78 MEN1 (0.47) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL12415529 0.74 ALDH1A1 (0.66) ALDH1A1MEN1KMT2ANPC1POLB
SCHEMBL8677385 0.72 ALDH1A1 (0.59) ALDH1A1RAB9AHTTACHELMNA
SCHEMBL7703726 0.69 S100A4 (0.44) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL28501723 0.69 CASP6 (0.43) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL29584495 0.67 HDAC3 (0.44) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL13621750 0.65 POLB (0.64) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL7706701 0.64 MEN1 (0.47) ALDH1A1MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed