SCHEMBL2852896

SCHEMBL2852896

O=C(NCc1ccccc1)c1cnn(-c2ccc(F)cc2)c1C(F)(F)F

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.63
ALDH1A1 P00352 2/20 0.63
CCR1 P32246 9/20 0.62
HPGD P15428 1/20 0.59
DDR1 Q08345 1/20 0.58
MAPK11 Q15759 1/20 0.58
MAPK14 Q16539 1/20 0.58
DDR2 Q16832 1/20 0.58
TMEM97 Q5BJF2 1/20 0.58
MAP3K20 Q9NYL2 1/20 0.58
MAP3K2 Q9Y2U5 1/20 0.58
MAPT P10636 3/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
POLB P06746 1/20 0.56
TP53 P04637 1/20 0.56
NPC1 O15118 1/20 0.53
HTT P42858 1/20 0.53
RAB9A P51151 1/20 0.53
SMO Q99835 1/20 0.53
MAPK1 P28482 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852102 0.95 ALDH1A1 (0.67) KDM4EALDH1A1CCR1HPGDDDR1
SCHEMBL2860213 0.93 KDM4E (0.73) KDM4EALDH1A1CCR1HPGDDDR1
SCHEMBL2850153 0.91 KDM4E (0.63) KDM4EALDH1A1CCR1HPGDDDR1
SCHEMBL2850548 0.90 CCR1 (0.61) KDM4EALDH1A1CCR1DDR1MAPK11
SCHEMBL2852015 0.90 CCR1 (0.63) KDM4EALDH1A1CCR1HPGDDDR1
SCHEMBL2856181 0.89 CCR1 (0.56) KDM4EALDH1A1CCR1DDR1MAPK11
SCHEMBL2859017 0.89 MAPT (0.69) KDM4EALDH1A1CCR1DDR1MAPK11
SCHEMBL2857342 0.89 CCR1 (0.60) KDM4EALDH1A1CCR1HPGDDDR1
SCHEMBL2856191 0.88 CCR1 (0.80) KDM4EALDH1A1CCR1
SCHEMBL2855115 0.87 CCR1 (0.64) KDM4EALDH1A1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed