SCHEMBL28503302

SCHEMBL28503302

CC(N)(Cc1ccc(COc2ccncc2)cc1)C(N)=O

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 4/20 0.45
BLM P54132 1/20 0.44
MAOB P27338 4/20 0.44
NR4A2 P43354 1/20 0.42
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
KDM1A O60341 1/20 0.41
RCOR1 Q9UKL0 1/20 0.41
MAPK14 Q16539 1/20 0.40
MMP2 P08253 1/20 0.40
MMP13 P45452 1/20 0.40
GPR119 Q8TDV5 1/20 0.40
EPHX2 P34913 1/20 0.39
PPARG P37231 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8935338 0.96 PARP10 (0.48) PARP10BLMMAOBNR4A2RXRA
SCHEMBL27344680 0.90 MMP13 (0.44) PARP10MAOBMAPK14MMP2MMP13
SCHEMBL28491503 0.87 PKM (0.45) PARP10MAOBALDH1A1RAB9AKDM1A
SCHEMBL27311683 0.86 PPARG (0.53) PARP10BLMMAOBNR4A2ALDH1A1
SCHEMBL28904310 0.84 NPC1 (0.56) PARP10MAOBALDH1A1POLBMAPT
SCHEMBL27309675 0.84 PARP10 (0.57) PARP10MAOBNR4A2MAPTRAB9A
SCHEMBL28505503 0.84 RAB9A (0.51) BLMALDH1A1MAPTRAB9AMMP2
SCHEMBL28510234 0.83 MAOB (0.57) PARP10MAOBNR4A2RAB9A
SCHEMBL28500733 0.83 MAOB (0.61) PARP10MAOBNR4A2
Hydrochloric Acid SCHEMBL27353104 0.83 PARP10 (0.56) PARP10MAOBNR4A2MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107522654-B Novel alpha-aminoamide derivatives and medicinal use thereof 中国人民解放军军事医学科学院毒物药物研究所 2020-09-01 CN disclosed