SCHEMBL2850346

SCHEMBL2850346

O=C(NCc1ccc2c(c1)OCO2)Oc1cnn(-c2cc(Cl)ccc2Cl)c1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.48
ALDH1A1 P00352 4/20 0.46
HTT P42858 2/20 0.46
HPGD P15428 2/20 0.46
LMNA P02545 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HEXD Q8WVB3 1/20 0.46
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
TRPV1 Q8NER1 2/20 0.44
TP53 P04637 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
TSHR P16473 1/20 0.43
POLB P06746 2/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856260 0.88 TSHR (0.46) SMN1; SMN2HPGDLMNATRPV1TSHR
SCHEMBL2857628 0.84 NPC1 (0.40) SMN1; SMN2ALDH1A1HPGDLMNATP53
SCHEMBL2857977 0.84 ALDH1A1 (0.47) SMN1; SMN2ALDH1A1HTTHPGDLMNA
SCHEMBL2848518 0.84 ALDH1A1 (0.58) SMN1; SMN2ALDH1A1HTTHPGDLMNA
SCHEMBL2855603 0.83 P2RX1 (0.44) HPGDLMNANPSR1POLB
SCHEMBL2861682 0.83 ALDH1A1 (0.48) SMN1; SMN2ALDH1A1HTTHPGDLMNA
SCHEMBL2856388 0.83 TRPV1 (0.51) SMN1; SMN2ALDH1A1HTTLMNAL3MBTL1
SCHEMBL2850129 0.83 ALDH1A1 (0.52) SMN1; SMN2ALDH1A1HTTHPGDCYP1A2
SCHEMBL2854686 0.83 SMN1; SMN2 (0.52) SMN1; SMN2ALDH1A1HTTHPGDL3MBTL1
SCHEMBL2852539 0.83 LMNA (0.52) HPGDLMNACYP1A2CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed