SCHEMBL2861682

SCHEMBL2861682

O=C(NCc1ccc2c(c1)OCO2)Oc1cnn(-c2cccc(Cl)n2)c1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.45
ALDH2 P05091 1/20 0.44
POLB P06746 2/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
HPGD P15428 4/20 0.43
TSHR P16473 2/20 0.43
TRPV1 Q8NER1 1/20 0.43
LMNA P02545 2/20 0.42
MAPK1 P28482 2/20 0.42
MMP13 P45452 1/20 0.42
KDM4E B2RXH2 2/20 0.42
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2857977 0.87 ALDH1A1 (0.47) ALDH1A1HTTSMN1; SMN2ALDH2POLB
SCHEMBL2852370 0.87 ALDH1A1 (0.52) ALDH1A1HTTSMN1; SMN2POLBKMT2A
SCHEMBL2848518 0.85 ALDH1A1 (0.58) ALDH1A1HTTSMN1; SMN2POLBMEN1
SCHEMBL2850129 0.84 ALDH1A1 (0.52) ALDH1A1HTTSMN1; SMN2POLBKMT2A
SCHEMBL2853347 0.84 TRPV1 (0.41) ALDH1A1HPGDTRPV1
SCHEMBL2850346 0.83 SMN1; SMN2 (0.48) ALDH1A1HTTSMN1; SMN2ALDH2POLB
SCHEMBL2856388 0.83 TRPV1 (0.51) ALDH1A1HTTSMN1; SMN2POLBMEN1
SCHEMBL2854686 0.83 SMN1; SMN2 (0.52) ALDH1A1HTTSMN1; SMN2POLBMEN1
SCHEMBL2852635 0.81 EPHX1 (0.44) MEN1KMT2AMAPK1
SCHEMBL2856620 0.81 ALDH1A1 (0.50) ALDH1A1HTTSMN1; SMN2POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed