SCHEMBL28503532

SCHEMBL28503532

C[Si](C)(C)CCOCn1cc(I)cc1Br

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.41
EGFR P00533 1/20 0.32
IGF1R P08069 1/20 0.32
SRC P12931 1/20 0.32
FLT4 P35916 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
EPHB4 P54760 1/20 0.32
TEK Q02763 1/20 0.32
PDE10A Q9Y233 2/20 0.30
KLKB1 P03952 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29112575 0.81 DGAT1 (0.41) DGAT1EGFRIGF1RSRCFLT4
SCHEMBL28562824 0.78 DGAT1 (0.40) DGAT1EGFRIGF1RSRCFLT4
SCHEMBL28645169 0.78 DGAT1 (0.39) DGAT1PDE10A
SCHEMBL23997682 0.77 KLKB1 (0.47) DGAT1EGFRIGF1RSRCFLT4
SCHEMBL21712951 0.75 KLKB1 (0.37) DGAT1EGFRIGF1RSRCFLT4
SCHEMBL4394992 0.74 DGAT1 (0.43) DGAT1PDE10AKLKB1
SCHEMBL17796240 0.74 ALDH1A1 (0.34) DGAT1EGFRIGF1RSRCFLT4
SCHEMBL29023457 0.73 DGAT1 (0.44) DGAT1EGFRIGF1RSRCFLT4
SCHEMBL27858492 0.73 DGAT1 (0.36) DGAT1EGFRIGF1RSRCFLT4
SCHEMBL4394623 0.73 DGAT1 (0.39) DGAT1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed