SCHEMBL23997682

SCHEMBL23997682

C[Si](C)(C)CCOCn1cc(I)cc1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.47
NPC1 O15118 1/20 0.37
DGAT1 O75907 6/20 0.34
EGFR P00533 1/20 0.32
IGF1R P08069 1/20 0.32
SRC P12931 1/20 0.32
FLT4 P35916 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
EPHB4 P54760 1/20 0.32
TEK Q02763 1/20 0.32
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21712951 0.86 KLKB1 (0.37) KLKB1NPC1DGAT1EGFRIGF1R
SCHEMBL17222119 0.83 KLKB1 (0.47) KLKB1NPC1DGAT1EGFRIGF1R
SCHEMBL25254975 0.83 KLKB1 (0.47) KLKB1NPC1DGAT1MAPT
SCHEMBL5654607 0.80 KLKB1 (0.45) KLKB1NPC1DGAT1
SCHEMBL28503532 0.77 DGAT1 (0.41) KLKB1NPC1DGAT1EGFRIGF1R
SCHEMBL17222067 0.74 KLKB1 (0.45) KLKB1NPC1DGAT1EGFRIGF1R
SCHEMBL12984274 0.74 KLKB1 (0.41) KLKB1NPC1DGAT1EGFRIGF1R
SCHEMBL29977642 0.74 KLKB1 (0.39) KLKB1NPC1DGAT1MAPT
SCHEMBL17796240 0.72 ALDH1A1 (0.34) NPC1DGAT1EGFRIGF1RSRC
SCHEMBL874860 0.72 GPR35 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922535-B1 THROMBIN INHIBITORS MERCK SHARP & DOHME (US) 2021-11-10 EP disclosed