SCHEMBL28504646

SCHEMBL28504646

CN(C)CCN(C)C(=O)c1ccc(B(O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.46
DRD2 P14416 1/20 0.42
PDK1 Q15118 1/20 0.41
MCHR1 Q99705 1/20 0.40
MLYCD O95822 1/20 0.39
ESRRG P62508 1/20 0.39
PDE7A Q13946 1/20 0.39
HDAC6 Q9UBN7 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
PIK3CA P42336 2/20 0.38
MTOR P42345 2/20 0.38
PIK3CG P48736 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28499683 0.90 HDAC6 (0.43) HDAC4DRD2MCHR1MLYCDESRRG
SCHEMBL26699702 0.86 NAMPT (0.46) DRD2MLYCDESRRGHDAC6LPL
SCHEMBL490705 0.82 LPL (0.44) HDAC4MLYCDLPLLIPG
SCHEMBL22858927 0.81 ALDH1A1 (0.50) MLYCD
SCHEMBL12237841 0.80 CDK4 (0.50) HDAC4DRD2PDK1MCHR1MLYCD
SCHEMBL25975198 0.80 HDAC4 (0.49) HDAC4DRD2PDK1MCHR1MLYCD
SCHEMBL177498 0.80 MLYCD (0.64) MCHR1MLYCDESRRG
SCHEMBL28513496 0.80 DRD2 (0.44) HDAC4DRD2MLYCDHDAC6HDAC3
SCHEMBL4022759 0.79 DPP4 (0.40) HDAC6HDAC1LPLLIPG
SCHEMBL15208211 0.79 HDAC4 (0.48) HDAC4DRD2PDK1MCHR1MLYCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed