SCHEMBL28508404

SCHEMBL28508404

O=S(=O)(Oc1cccc2c(N3CCOCC3)c(N3CCOCC3)cnc12)C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.45
TP53 P04637 1/20 0.45
MAPK1 P28482 1/20 0.45
RECQL P46063 1/20 0.45
HSD17B10 Q99714 1/20 0.45
SLC6A3 Q01959 1/20 0.38
SLC40A1 Q9NP59 1/20 0.37
PIK3CB P42338 1/20 0.37
MAPT P10636 3/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
GLA P06280 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PRKDC P78527 2/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28511308 0.85 SLC40A1 (0.47) SLC40A1PIK3CBMAPTHTTPRKDC
SCHEMBL28518634 0.77 KDM4E (0.44) PIK3CBKDM4E
SCHEMBL2198567 0.76 MAPT (0.53) MAPTLMNANPSR1POLB
SCHEMBL31239122 0.75 DRD2 (0.42) PIK3CBMAPTLMNAPRKDCPOLB
SCHEMBL1275376 0.70 PRKDC (0.58) PIK3CBPRKDC
SCHEMBL434090 0.69 PRKDC (0.67) TP53HSD17B10PIK3CBKDM4ELMNA
SCHEMBL13403537 0.68 PIK3CG (0.64) PIK3CBKDM4EPRKDC
SCHEMBL15125330 0.67 DRD2 (0.35)
SCHEMBL2197587 0.67 KMO (0.51) LMNAHTTPRKDC
SCHEMBL31156589 0.66 KDM4E (0.43) MAPK1HSD17B10SLC40A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300126-A Heterocyclic DNA-PK inhibitors 山东轩竹医药科技有限公司 2021-02-02 CN disclosed