SCHEMBL28508807

SCHEMBL28508807

COc1ccc2oc(=O)c(C(=O)CBr)cc2c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.71
ALDH1A1 P00352 5/20 0.71
HPGD P15428 2/20 0.71
CA12 O43570 1/20 0.71
CA1 P00915 1/20 0.71
CA2 P00918 1/20 0.71
CA3 P07451 1/20 0.71
CA6 P23280 1/20 0.71
CA5A P35218 1/20 0.71
CA7 P43166 1/20 0.71
CA9 Q16790 1/20 0.71
CA14 Q9ULX7 1/20 0.71
CA5B Q9Y2D0 1/20 0.71
MAOB P27338 5/20 0.67
GAA P10253 3/20 0.66
KMT2A Q03164 1/20 0.61
MAPT P10636 2/20 0.60
GLA P06280 1/20 0.60
CYP2C19 P33261 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2032914 0.84 KDM4E (0.81) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL7527810 0.83 ALDH1A1 (1.00) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL29963204 0.83 KDM4E (1.00) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL978456 0.83 KDM4E (1.00) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL28703856 0.82 MAOB (0.68) CA12CA1CA2CA6CA5A
SCHEMBL8310947 0.82 TAS1R3 (0.59) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL6835643 0.82 KDM4E (0.76) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL28690050 0.80 MAOA (0.68) KDM4ECA12CA1CA2CA3
SCHEMBL2031783 0.80 MAOB (1.00) KDM4EALDH1A1HPGDCA12CA1
SCHEMBL12838815 0.80 KDM4E (1.00) KDM4EALDH1A1HPGDCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108774277-B Thiazole derivative containing glucosamine and coumarin molecules, and preparation method and application thereof 淮海工学院 2021-12-21 CN disclosed
CN-108558843-B Coumarin-triazole-isatin type compound and preparation method and application thereof 贵州医科大学 2020-12-15 CN disclosed