SCHEMBL28513499

SCHEMBL28513499

CCOC(=O)c1nn(CC)c(Cl)c1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 3/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
PDE4A P27815 7/20 0.46
PDE4B Q07343 7/20 0.46
PDE4C Q08493 7/20 0.46
PDE4D Q08499 7/20 0.46
KMT2A Q03164 1/20 0.42
CYP1A2 P05177 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
APP P05067 1/20 0.40
MAPT P10636 1/20 0.40
CASP1 P29466 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1996657 0.77 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHSD17B10PDE4A
SCHEMBL3382168 0.74 KMT2A (0.44) ALDH1A1HPGDPDE4APDE4BPDE4C
SCHEMBL22900713 0.73 PDE4A (0.47) ALDH1A1KDM4EPDE4APDE4BPDE4C
SCHEMBL22609267 0.72 MAPK1 (0.62) ALDH1A1KDM4EHPGDHSD17B10PDE4A
SCHEMBL22900339 0.71 PDE4A (0.45) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL29031589 0.71 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHSD17B10PDE4D
SCHEMBL32663296 0.70 SMN1; SMN2 (0.42) ALDH1A1KDM4EPDE4APDE4BPDE4C
SCHEMBL14304442 0.69 ADORA3 (0.47) ALDH1A1KDM4EHPGDHSD17B10KMT2A
SCHEMBL30685706 0.69 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDHSD17B10PDE4A
SCHEMBL2843820 0.68 ALDH1A1 (0.59) ALDH1A1KDM4EHPGDHSD17B10KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108431004-B Heterocyclic compounds 武田药品工业株式会社 2021-02-12 CN disclosed