SCHEMBL28513873

SCHEMBL28513873

COc1cc(Br)cc(OC)c1N1CCN(C)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
DRD2 P14416 2/20 0.47
DRD3 P35462 2/20 0.47
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
CCR4 P51679 1/20 0.43
HTR6 P50406 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
HTR1A P08908 1/20 0.42
CYP2D6 P10635 1/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR1E P28566 1/20 0.42
HTR1F P30939 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTR7 P34969 1/20 0.42
ADRA1B P35368 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21590338 0.90 GAA (0.47) GAADRD2DRD3MAPTMAPK1
SCHEMBL21590174 0.89 GAA (0.46) GAADRD2DRD3MAPTMAPK1
SCHEMBL5240485 0.85 KDM4E (0.46) GAAMAPTHTR2A
SCHEMBL28503601 0.85 ALDH1A1 (0.41) GAADRD2HTR1AADRA1B
SCHEMBL28511352 0.80 CHRNB2 (0.53) DRD2DRD3MAPTHTR6HTR1A
SCHEMBL21388456 0.80 MAPT (0.43) GAADRD2DRD3MAPTMAPK1
SCHEMBL2799605 0.77 DRD2 (0.60) GAADRD2DRD3MAPTMAPK1
SCHEMBL21388389 0.76 MAPT (0.46) DRD2DRD3MAPTCCR4HTR1A
SCHEMBL21388463 0.75 DRD2 (0.45) DRD2DRD3MAPTCCR4HTR1A
SCHEMBL17310109 0.75 ACHE (0.50) GAADRD2DRD3CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed