SCHEMBL28514129

SCHEMBL28514129

c1ccc(CN2CCC(COc3cncc(-n4cccc4)c3)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.51
GSK3B P49841 2/20 0.51
MAOA P21397 2/20 0.50
MAOB P27338 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28512442 0.84 ACHE (0.53) ACHEGSK3BMAOAMAOB
SCHEMBL29960864 0.84 ACHE (0.53) ACHEGSK3BMAOAMAOB
SCHEMBL8549837 0.79 CCR3 (0.63)
Hydrochloric Acid SCHEMBL8681764 0.77 CCR3 (0.61)
SCHEMBL7520395 0.77 CHRNB2 (0.55) ACHEGSK3BMAOAMAOB
SCHEMBL7521464 0.77 ACHE (0.52) ACHEGSK3BMAOAMAOB
SCHEMBL7520899 0.77 CHRNB2 (0.47) ACHEGSK3BMAOAMAOB
SCHEMBL12192898 0.75 ROCK1 (0.61) ACHEMAOAMAOB
SCHEMBL7330801 0.74 SLC6A2 (0.60) ACHEMAOAMAOB
SCHEMBL7296120 0.74 ALDH1A1 (0.65) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112047928-A Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2020-12-08 CN claimed
CN-112047928-B Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2022-09-23 CN disclosed
CN-112047928-A Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2020-12-08 CN disclosed