SCHEMBL28514488

SCHEMBL28514488

Cc1cccc(CN2CCN(C=O)CC2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.58
KDM4E B2RXH2 4/20 0.58
HTT P42858 2/20 0.58
FAAH O00519 1/20 0.56
MAPT P10636 1/20 0.56
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
LMNA P02545 1/20 0.53
ACHE P22303 1/20 0.52
USP2 O75604 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
HPN P05981 1/20 0.52
CHRM2 P08172 1/20 0.52
ADRA2A P08913 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
CHRM1 P11229 1/20 0.52
DRD2 P14416 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30463522 1.00 ALDH1A1 (0.58) ALDH1A1KDM4EHTTFAAHMAPT
SCHEMBL1134938 0.81 SIGMAR1 (0.72) ALDH1A1KMT2ALMNADRD4
SCHEMBL7428714 0.81 SIGMAR1 (0.76) ALDH1A1KDM4EHTTFAAHMAPT
SCHEMBL7426490 0.81 ALDH1A1 (0.64) ALDH1A1KDM4EFAAHMEN1KMT2A
SCHEMBL2325343 0.80 LMNA (0.68) ALDH1A1KDM4EFAAHMAPTMEN1
SCHEMBL15829984 0.80 ALDH1A1 (0.62) ALDH1A1KDM4EHTTFAAHMAPT
SCHEMBL10076573 0.80 MC4R (0.65) ALDH1A1KDM4EHTTFAAHMAPT
SCHEMBL31546411 0.80 HRH3 (0.69) ALDH1A1KDM4EHTTMAPT
SCHEMBL12981 0.80 HRH3 (0.69) ALDH1A1KDM4EHTTMAPT
SCHEMBL5542258 0.79 FAAH (0.54) ALDH1A1FAAHKMT2ALMNADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300145-B Tri-aromatic ring compound targeting STAT3 bifunctional phosphorylation site and application thereof 上海宇耀生物科技有限公司 2023-07-21 CN claimed
CN-112300145-A Three-aromatic ring compound targeting STAT3 bifunctional phosphorylation site and application thereof 上海宇耀生物科技有限公司 2021-02-02 CN claimed
CN-117986254-A Hirsutine alkaloid derivative, and preparation method and application thereof 中国海洋大学 2024-05-07 CN disclosed
CN-112300145-B Tri-aromatic ring compound targeting STAT3 bifunctional phosphorylation site and application thereof 上海宇耀生物科技有限公司 2023-07-21 CN disclosed
CN-112300145-A Three-aromatic ring compound targeting STAT3 bifunctional phosphorylation site and application thereof 上海宇耀生物科技有限公司 2021-02-02 CN disclosed