SCHEMBL285168

SCHEMBL285168

C(=C/c1ccccc1-c1nc2ccccc2o1)\c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.48
MAPT P10636 6/20 0.48
HPGD P15428 5/20 0.48
KDM4E B2RXH2 5/20 0.48
USP2 O75604 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
TOP2A P11388 1/20 0.47
NPC1 O15118 6/20 0.46
RAB9A P51151 6/20 0.46
HSD17B10 Q99714 4/20 0.46
TP53 P04637 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
PKM P14618 2/20 0.46
GAA P10253 2/20 0.46
GLA P06280 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
KDM6B O15054 1/20 0.46
KDM6A O15550 1/20 0.46
KMT2A Q03164 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28887970 1.00 ALDH1A1 (0.48) ALDH1A1MAPTHPGDKDM4EUSP2
SCHEMBL285170 1.00 ALDH1A1 (0.48) ALDH1A1MAPTHPGDKDM4EUSP2
SCHEMBL11447095 0.94 ALDH1A1 (0.46) ALDH1A1MAPTHPGDKDM4EUSP2
SCHEMBL11458764 0.94 ALDH1A1 (0.46) ALDH1A1MAPTHPGDKDM4EUSP2
SCHEMBL250148 0.92 TOP2A (0.53) ALDH1A1MAPTHPGDKDM4EUSP2
SCHEMBL22687002 0.92 TOP2A (0.53) ALDH1A1MAPTHPGDKDM4EUSP2
SCHEMBL5335888 0.92 TOP2A (0.53) ALDH1A1MAPTHPGDKDM4EUSP2
SCHEMBL250150 0.89 TOP2A (0.46) ALDH1A1MAPTHPGDKDM4EUSP2
SCHEMBL19717967 0.89 TOP2A (0.46) ALDH1A1MAPTHPGDKDM4EUSP2
SCHEMBL7567677 0.88 PTGS2 (0.50) ALDH1A1MAPTHPGDKDM4EUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 361 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10254646-B2 Composition sensitive to radiation in electromagnetic spectrum ranges for printing purposes, printing plate comprising said composition, use of said composition and image development process IBF INDUSTRIA BRASILEIRA DE FILMES S/A (BR) 2019-04-09 US claimed
US-20160026080-A1 COMPOSITION SENSITIVE TO RADIATION IN ELECTROMAGNETIC SPECTRUM RANGES FOR PRINTING PURPOSES, PRINTING PLATE COMPRISING SAID COMPOSITION, USE OF SAID COMPOSITION AND IMAGE DEVLOPMENT PROCESS IBF INDUSTRIA BRASILEIRA DE FILMES S/A (BR) 2016-01-28 US claimed
EP-2937733-A1 COMPOSITION SENSITIVE TO RADIATION IN ELECTROMAGNETIC SPECTRUM RANGES FOR PRINTING PURPOSES, PRINTING PLATE COMPRISING SAID COMPOSITION, USE OF SAID COMPOSITION AND IMAGE DEVELOPMENT PROCESS IBF - Indústria Brasileira de Filmes S/A (BR) 2015-10-28 EP claimed
EP-1531170-B1 Ultraviolet blocking composition for protection of package or container contents EASTMAN CHEM CO (US) 2014-10-29 EP claimed
EP-1965231-A2 Optical Diffuser Film and Light Assembly for liquid crystal displays Rohm and Haas Denmark Finance A/S (DK) 2008-09-03 EP claimed
US-20080192352-A1 Optical diffuser film and light assembly EASTMAN KODAK COMPANY 2008-08-14 US claimed
EP-1848763-B1 MOULDED OBJECT EXHIBITING A POLYCHROMATIC EFFECT, ASSOCIATED LIGHT DEVICE AND RESIN ARKEMA FRANCE (FR) 2008-04-16 EP claimed
EP-1848763-A1 MOULDED OBJECT EXHIBITING A POLYCHROMATIC EFFECT, ASSOCIATED LIGHT DEVICE AND RESIN Arkema France (FR) 2007-10-31 EP claimed
US-7157547-B2 Ultraviolet blocking composition for protection of package or container contents EASTMAN CHEMICAL COMPANY (US) 2007-01-02 US claimed
EP-1325067-B1 MULTI-COMPONENT OPTICALLY BRIGHTENED POLYOLEFIN BLEND EASTMAN CHEM CO (US) 2006-09-06 EP claimed
EP-0020298-B1 BENZOXAZOLYL STILBENES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS OPTICAL BRIGHTENERS FOR ORGANIC MATERIALS CIBA-GEIGY AG (CH) 1983-06-22 EP claimed
EP-0017618-B1 PROCESS FOR OPTICALLY BRIGHTENING POLYESTER FIBRES BY THE EXHAUST PROCESS CIBA-GEIGY AG (CH) 1983-03-02 EP claimed
EP-0054511-A2 4-Styryl-4'-vinylbifenyls, methods for their preparation and their use as optical whiteners CIBA-GEIGY AG (CH) 1982-06-23 EP claimed
US-4297234-A OPTICAL BRIGHTENERS CIBA-GEIGY CORPORATION (US) 1981-10-27 US claimed
EP-0033459-A1 Benzoxazolylstilbenes, processes for their production and their use as optical brighteners BAYER AG (DE) 1981-08-12 EP claimed
US-4283197-A Process for whitening polyester fibres by the exhaust method CIBA-GEIGY CORPORATION (US) 1981-08-11 US claimed
EP-0030917-A2 Optical brighteners from bistyryl benzene, process for their preparation and their use CIBA-GEIGY AG (CH) 1981-06-24 EP claimed
EP-0020298-A1 Benzoxazolyl stilbenes, process for their preparation and their use as optical brighteners for organic materials CIBA-GEIGY AG (CH) 1980-12-10 EP claimed
US-4036778-A Aqueous, storage-stable dispersions of water-soluble compounds CIBA-GEIGY CORPORATION (US) 1977-07-19 US claimed
US-3996210-A OPTICAL BRIGHTENERS SANDOZ LTD. (CH) 1976-12-07 US claimed