SCHEMBL28518969

SCHEMBL28518969

NC(=O)Oc1ccc(Oc2ccnc(N)c2N)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MET P08581 19/20 0.41
KDR P35968 2/20 0.41
RET P07949 1/20 0.41
KIT P10721 1/20 0.41
PDGFRA P16234 1/20 0.41
FLT3 P36888 1/20 0.41
CYP3A4 P08684 3/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2934749 0.90 MET (0.40) METKDRRETKITPDGFRA
SCHEMBL28529335 0.83 MAPT (0.41) METKDRRETKITPDGFRA
SCHEMBL23070954 0.83 MET (0.39) METKDRRETKITPDGFRA
SCHEMBL29148908 0.79 MET (0.43) METKDRRETKITPDGFRA
SCHEMBL2934893 0.76 MET (0.54) METKDRRETKITPDGFRA
SCHEMBL3759422 0.76 MET (0.38) METKDRRETKITPDGFRA
SCHEMBL28524104 0.75 BRAF (0.52)
SCHEMBL23070949 0.75 BRAF (0.53)
SCHEMBL2935339 0.74 PDGFRB (0.34) METKDRPDGFRA
SCHEMBL6032672 0.74 MET (0.52) MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116283916-B Compound with Axl and c-Met kinase inhibition activity and preparation and application thereof 中国科学院上海药物研究所 2024-06-11 CN disclosed
CN-117500805-A Novel urea derivative compounds as RON inhibitors 株式会社LG化学 2024-02-02 CN disclosed
CN-117500804-A Novel urea derivative compounds as RON inhibitors 株式会社LG化学 2024-02-02 CN disclosed
CN-116283916-A Compound with Axl and c-Met kinase inhibition activity and preparation and application thereof 中国科学院上海药物研究所 2023-06-23 CN disclosed
CN-112457295-B Compound with Axl and c-Met kinase inhibitory activity and preparation and application thereof 中国科学院上海药物研究所 2022-07-26 CN disclosed
CN-112457295-A Compound with Axl and c-Met kinase inhibitory activity and preparation and application thereof 中国科学院上海药物研究所 2021-03-09 CN disclosed