SCHEMBL2851983

SCHEMBL2851983

CCN(Cc1cccs1)C(=O)c1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.61
NPSR1 Q6W5P4 2/20 0.61
HSP90AA1 P07900 1/20 0.61
MAPK1 P28482 1/20 0.61
TRPM8 Q7Z2W7 5/20 0.49
MAPT P10636 4/20 0.45
GPR6 P46095 1/20 0.43
POLB P06746 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 1/20 0.42
KDM4E B2RXH2 1/20 0.41
UBE2M P61081 1/20 0.41
DCUN1D1 Q96GG9 1/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
NR3C1 P04150 1/20 0.41
TRPC3 Q13507 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852994 0.89 ALDH1A1 (0.56) ALDH1A1NPSR1HSP90AA1MAPK1TRPM8
SCHEMBL10366449 0.86 MAPT (0.53) ALDH1A1NPSR1HSP90AA1MAPK1MAPT
SCHEMBL2854667 0.84 ALDH1A1 (0.55) ALDH1A1NPSR1HSP90AA1MAPK1MAPT
SCHEMBL2852358 0.83 ALDH1A1 (0.48) ALDH1A1NPSR1HSP90AA1MAPK1MAPT
SCHEMBL2856206 0.83 ALDH1A1 (0.48) ALDH1A1NPSR1HSP90AA1MAPK1MAPT
SCHEMBL2852819 0.82 CCR1 (0.57) ALDH1A1NPSR1HSP90AA1MAPK1MAPT
SCHEMBL16615747 0.82 ALDH1A1 (0.65) ALDH1A1NPSR1HSP90AA1MAPK1TRPM8
SCHEMBL2862176 0.79 TRPV1 (0.47) ALDH1A1NPSR1HSP90AA1MAPK1MAPT
SCHEMBL10365422 0.77 MAPT (0.67) ALDH1A1MAPTPOLBSMN1; SMN2LMNA
SCHEMBL10366936 0.77 KEAP1 (0.52) ALDH1A1MAPTPOLBSMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed