SCHEMBL2852082

SCHEMBL2852082

COc1ccc(-n2ncc(C(=O)NCc3ccc(Cl)cc3)c2C)cc1

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 5/20 0.72
HPGD P15428 2/20 0.63
ABCB1 P08183 1/20 0.58
LMNA P02545 3/20 0.57
MAPT P10636 2/20 0.57
NPSR1 Q6W5P4 1/20 0.56
NPC1 O15118 1/20 0.55
PKM P14618 1/20 0.55
RAB9A P51151 1/20 0.55
NR3C1 P04150 1/20 0.55
PDE2A O00408 1/20 0.54
RXFP1 Q9HBX9 2/20 0.54
TP53 P04637 3/20 0.54
ALDH1A1 P00352 1/20 0.52
CYP1A1 P04798 1/20 0.50
LSS P48449 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855676 0.89 CCR1 (0.63) CCR1HPGDMAPTNPSR1NPC1
SCHEMBL2857166 0.89 HPGD (0.80) CCR1HPGDMAPTNPC1PKM
SCHEMBL2857860 0.87 CCR1 (0.75) CCR1HPGDMAPTNPSR1ALDH1A1
SCHEMBL2850617 0.86 HPGD (0.84) CCR1HPGDNPSR1NPC1PKM
SCHEMBL2859678 0.85 CCR1 (0.55) CCR1ABCB1LMNAMAPTNR3C1
SCHEMBL2854531 0.83 LMNA (0.52) CCR1ABCB1LMNAMAPTNPC1
SCHEMBL2856505 0.83 TP53 (0.59) CCR1HPGDLMNAMAPTNPSR1
SCHEMBL2850603 0.80 HPGD (0.73) CCR1HPGDMAPTNPSR1NPC1
SCHEMBL2859795 0.79 NPC1 (0.59) CCR1HPGDLMNAMAPTNPSR1
SCHEMBL2851942 0.78 NPC1 (0.64) HPGDMAPTNPC1PKMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed