SCHEMBL2859795

SCHEMBL2859795

COc1ccc(-n2ncc(C(=O)NCc3ccccc3F)c2C)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.59
RAB9A P51151 4/20 0.59
PKM P14618 1/20 0.59
HPGD P15428 3/20 0.57
MAPT P10636 5/20 0.54
NFKB1 P19838 1/20 0.54
NFKB2 Q00653 1/20 0.54
RELA Q04206 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
POLB P06746 2/20 0.53
CCR1 P32246 2/20 0.51
ALDH1A1 P00352 3/20 0.49
TP53 P04637 1/20 0.48
GAA P10253 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
LMNA P02545 1/20 0.48
EED O75530 1/20 0.48
RBBP4 Q09028 1/20 0.48
SUZ12 Q15022 1/20 0.48
EZH2 Q15910 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852886 0.89 CCR1 (0.62) NPC1RAB9AHPGDMAPTPOLB
SCHEMBL2854454 0.89 HPGD (0.72) NPC1RAB9APKMHPGDMAPT
SCHEMBL2856505 0.88 TP53 (0.59) NPC1RAB9APKMHPGDMAPT
SCHEMBL2857166 0.85 HPGD (0.80) NPC1RAB9APKMHPGDMAPT
SCHEMBL2857338 0.84 RAB9A (0.47) NPC1RAB9APKMHPGDMAPT
SCHEMBL2855676 0.83 CCR1 (0.63) NPC1RAB9APKMHPGDMAPT
SCHEMBL2852637 0.79 NR3C1 (0.64) NPC1RAB9APKMHPGDMAPT
SCHEMBL2852082 0.79 CCR1 (0.72) NPC1RAB9APKMHPGDMAPT
SCHEMBL2851942 0.79 NPC1 (0.64) NPC1RAB9APKMHPGDMAPT
SCHEMBL2857152 0.77 NPC1 (0.91) NPC1RAB9APKMHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed