SCHEMBL2857166

SCHEMBL2857166

COc1ccc(-n2ncc(C(=O)NCc3ccccc3)c2C)cc1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.80
NPC1 O15118 4/20 0.67
RAB9A P51151 4/20 0.67
PKM P14618 1/20 0.67
MAPT P10636 2/20 0.61
NFKB1 P19838 1/20 0.61
NFKB2 Q00653 1/20 0.61
RELA Q04206 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
TP53 P04637 3/20 0.60
CCR1 P32246 6/20 0.57
NR3C1 P04150 1/20 0.56
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
PDE2A O00408 1/20 0.53
EED O75530 1/20 0.53
RBBP4 Q09028 1/20 0.53
SUZ12 Q15022 1/20 0.53
EZH2 Q15910 1/20 0.53
AEBP2 Q6ZN18 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856089 0.89 HPGD (1.00) HPGDNPC1RAB9APKMNFKB1
SCHEMBL2852082 0.89 CCR1 (0.72) HPGDNPC1RAB9APKMMAPT
SCHEMBL2855676 0.89 CCR1 (0.63) HPGDNPC1RAB9APKMMAPT
SCHEMBL2851942 0.89 NPC1 (0.64) HPGDNPC1RAB9APKMMAPT
SCHEMBL2854347 0.86 HPGD (0.84) HPGDNPC1RAB9AMAPTTP53
SCHEMBL2856505 0.85 TP53 (0.59) HPGDNPC1RAB9APKMMAPT
SCHEMBL2859795 0.85 NPC1 (0.59) HPGDNPC1RAB9APKMMAPT
SCHEMBL2850316 0.85 TP53 (0.59) HPGDMAPTSMN1; SMN2TP53CCR1
SCHEMBL2857152 0.82 NPC1 (0.91) HPGDNPC1RAB9APKMMAPT
SCHEMBL2860234 0.82 HPGD (0.54) HPGDNPC1RAB9APKMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed