SCHEMBL28522207

SCHEMBL28522207

C=CC(=O)Nc1ccc(OCCOC)nc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.61
ITK Q08881 4/20 0.61
TGM2 P21980 1/20 0.49
BTK Q06187 3/20 0.48
JAK2 O60674 1/20 0.48
LYN P07948 1/20 0.48
TEC P42680 1/20 0.48
TXK P42681 1/20 0.48
BMX P51813 1/20 0.48
JAK3 P52333 1/20 0.48
CD69 Q07108 1/20 0.48
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
MAPT P10636 2/20 0.47
KDM4E B2RXH2 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
LMNA P02545 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CXCR1 P25024 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28524018 0.87 EGFR (0.49) EGFRITKTGM2NPC1RAB9A
SCHEMBL28519662 0.86 EGFR (0.50) EGFRITKTGM2NPC1RAB9A
SCHEMBL4197685 0.84 RAB9A (0.63) EGFRITKTGM2NPC1RAB9A
SCHEMBL27961476 0.83 KMT2A (0.51) NPC1RAB9AMAPTKDM4EMEN1
SCHEMBL28310060 0.80 TGM2 (0.67) EGFRITKTGM2BTKJAK2
SCHEMBL14791196 0.80 EGFR (0.74) EGFRITKBTKJAK2LYN
SCHEMBL28463718 0.80 EGFR (0.63) EGFRITKTGM2BTKJAK2
SCHEMBL12519520 0.78 EGFR (1.00) EGFRITKBTKJAK2LYN
SCHEMBL28450293 0.77 EGFR (0.58) EGFRITKTGM2BTKJAK2
SCHEMBL28455574 0.77 EGFR (0.58) EGFRITKTGM2BTKJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409360-B Heteroaryl vinyl xanthine derivatives and uses thereof 广东东阳光药业有限公司 2022-12-23 CN disclosed
CN-112409360-A Heteroaryl vinyl xanthine derivatives and uses thereof 广东东阳光药业有限公司 2021-02-26 CN disclosed