SCHEMBL28524205

SCHEMBL28524205

OC1CCc2ccc(-c3ccccc3)nc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
TRPV1 Q8NER1 1/20 0.36
ACHE P22303 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
MAP2K3 P46734 1/20 0.35
ADORA1 P30542 3/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA2A P29274 2/20 0.35
GFRA3 O60609 1/20 0.35
RET P07949 1/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
ASIC3 Q9UHC3 1/20 0.34
RIPK1 Q13546 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28524204 1.00 MEN1 (0.44) MEN1RAB9AKMT2ATRPV1ACHE
SCHEMBL31598495 1.00 MEN1 (0.44) MEN1RAB9AKMT2ATRPV1ACHE
SCHEMBL14884989 0.90 ACHE (0.43) MEN1RAB9AKMT2AACHEALDH1A1
SCHEMBL3311055 0.90 ACHE (0.43) MEN1RAB9AKMT2AACHEALDH1A1
SCHEMBL10287024 0.90 ACHE (0.43) MEN1RAB9AKMT2AACHEALDH1A1
SCHEMBL31598496 0.89 RAB9A (0.40) MEN1RAB9AKMT2AACHEALDH1A1
SCHEMBL10286368 0.89 RAB9A (0.40) MEN1RAB9AKMT2AACHEALDH1A1
SCHEMBL11519752 0.74 RAB9A (0.37) MEN1RAB9AKMT2AALDH1A1ADORA1
SCHEMBL3311297 0.74 IRAK4 (0.46) MEN1RAB9AKMT2AALDH1A1MAP2K3
SCHEMBL11643241 0.73 MEN1 (0.48) MEN1RAB9AKMT2AALDH1A1MAP2K3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112521419-A Method for preparing chiral nitrogen-phosphorus ligand L-8 containing pyridocyclopentane 南京艾普特生物医药有限公司 2021-03-19 CN disclosed
CN-112521420-A Method for synthesizing chiral nitrogen and phosphorus ligand L-8 containing pyridocycloheptane 南京艾普特生物医药有限公司 2021-03-19 CN disclosed
CN-112375101-A Method for preparing chiral nitrogen-phosphorus ligand L-8 containing pyridocyclohexane 南京艾普特生物医药有限公司 2021-02-19 CN disclosed