SCHEMBL2852450

SCHEMBL2852450

O=C1c2ccccc2OCC1(Cl)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.42
TSHR P16473 1/20 0.42
CYP19A1 P11511 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 1/20 0.37
MAOB P27338 2/20 0.36
KMT2A Q03164 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
MEN1 O00255 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
CFTR P13569 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2107486 0.77 TSHR (0.42) PKMTSHRCYP19A1ALDH1A1MAPT
SCHEMBL2025120 0.77 PKM (0.42) PKMTSHRCYP19A1ALDH1A1MAPT
SCHEMBL2856269 0.73 PKM (0.39) PKMTSHRCYP19A1ALDH1A1MAPT
SCHEMBL571667 0.72 CYP19A1 (0.41) CYP19A1ALDH1A1MAPTHPGDMAOB
SCHEMBL9136839 0.72 PKM (0.47) PKMTSHRCYP19A1ALDH1A1MAOB
SCHEMBL4618755 0.72 TSHR (0.47) PKMTSHRCYP19A1ALDH1A1MAOB
SCHEMBL29448029 0.72 PKM (0.47) PKMTSHRCYP19A1ALDH1A1MAPT
SCHEMBL4618757 0.72 TSHR (0.47) PKMTSHRCYP19A1ALDH1A1MAOB
SCHEMBL1133012 0.72 PKM (0.47) PKMTSHRCYP19A1ALDH1A1MAPT
SCHEMBL149892 0.69 ALDH1A1 (0.37) PKMTSHRALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010042933-A9 INHIBITION AND TREATMENT OF PROSTATE CANCER METASTASIS NORTHWESTERN UNIVERSITY (US) 2010-07-08 WO disclosed
WO-2010042933-A2 INHIBITION AND TREATMENT OF PROSTATE CANCER METASTASIS NORTHWESTERN UNIVERSITY (US) 2010-04-15 WO disclosed
WO-2009049214-A2 INHIBITION AND TREATMENT OF PROSTATE CANCER METASTASIS NORTHWESTERN UNIVERSITY (US) 2009-04-16 WO disclosed