SCHEMBL28524920

SCHEMBL28524920

CC(C)(C)OC(=O)Nc1cccc(CC(O)c2nccs2)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.44
RPS6KB1 P23443 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.43
METAP1 P53582 1/20 0.43
CYP17A1 P05093 2/20 0.41
GLS O94925 1/20 0.41
HDAC3 O15379 4/20 0.40
HDAC1 Q13547 4/20 0.40
HDAC2 Q92769 4/20 0.40
HDAC8 Q9BY41 4/20 0.40
HDAC10 Q969S8 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
IDO1 P14902 1/20 0.40
PRMT5 O14744 1/20 0.39
WDR77 Q9BQA1 1/20 0.39
SREBF2 Q12772 1/20 0.39
NPY1R P25929 1/20 0.39
BRD4 O60885 1/20 0.39
NAMPT P43490 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29643010 1.00 AURKA (0.44) AURKARPS6KB1SIRT2METAP1CYP17A1
SCHEMBL29642984 0.90 AURKA (0.45) AURKARPS6KB1SIRT2METAP1CYP17A1
SCHEMBL28531300 0.90 AURKA (0.45) AURKARPS6KB1SIRT2METAP1CYP17A1
SCHEMBL23682527 0.90 AURKA (0.45) AURKARPS6KB1SIRT2METAP1CYP17A1
SCHEMBL29642978 0.85 METAP1 (0.40) AURKARPS6KB1SIRT2METAP1CYP17A1
SCHEMBL21598768 0.83 MAPT (0.43) AURKA
SCHEMBL21598770 0.83 MAPT (0.43) AURKA
SCHEMBL28524919 0.77 CTSA (0.40)
SCHEMBL27554182 0.77 SLC7A5 (0.46) AURKARPS6KB1SIRT2CYP17A1HDAC3
SCHEMBL7609410 0.75 L3MBTL1 (0.44) METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112437675-A Antibody drug conjugates for ablating hematopoietic stem cells 诺华股份有限公司 2021-03-02 CN disclosed