SCHEMBL2852545

SCHEMBL2852545

COc1ccc(-n2ncc(OC(=O)NCc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2C(F)(F)F)cc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 2/20 0.42
MCHR1 Q99705 1/20 0.42
CCR1 P32246 6/20 0.42
RECQL P46063 1/20 0.41
HPGD P15428 3/20 0.41
SMO Q99835 1/20 0.41
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 1/20 0.40
USP2 O75604 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
TP53 P04637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MAPK1 P28482 1/20 0.39
FAAH O00519 1/20 0.39
NTRK1 P04629 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854330 0.92 CCR1 (0.52) CCR1RECQLUSP2POLBFAAH
SCHEMBL2857994 0.91 MTOR (0.46) CCR1ALDH1A1KDM4ENPSR1
SCHEMBL2863210 0.89 CCR1 (0.50) CCR1SMOKDM4ENPSR1MAPK1
SCHEMBL2852520 0.88 TP53 (0.47) HPGDALDH1A1KDM4EPOLBGAA
SCHEMBL2853270 0.88 CCR1 (0.51) CCR1NPSR1
SCHEMBL2857073 0.88 CCR1 (0.48) CCR1ALDH1A1KDM4EPOLB
SCHEMBL2860466 0.87 RCE1 (0.47) CCR1SMOALDH1A1POLBGAA
SCHEMBL2856797 0.86 P2RX7 (0.45) CCR1SMOALDH1A1MAPK1
SCHEMBL2848661 0.86 ABCB1 (0.48) NPBWR1CCR1ALDH1A1POLBTP53
SCHEMBL2856625 0.86 TSHR (0.48) NPBWR1CCR1SMONPSR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed