SCHEMBL2856797

SCHEMBL2856797

COc1cc(CNC(=O)Oc2cnn(-c3ccc(F)cc3)c2C(F)(F)F)cc(OC)c1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.45
CCR1 P32246 6/20 0.44
SMO Q99835 8/20 0.43
ALDH1A1 P00352 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPK1 P28482 1/20 0.39
TRPA1 O75762 1/20 0.38
NR3C1 P04150 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853277 0.92 CCR1 (0.50) P2RX7CCR1SMO
SCHEMBL2855623 0.91 CCR1 (0.44) P2RX7CCR1SMO
SCHEMBL2860466 0.91 RCE1 (0.47) P2RX7CCR1SMOALDH1A1L3MBTL1
SCHEMBL2850314 0.91 P2RX7 (0.42) P2RX7CCR1SMOALDH1A1L3MBTL1
SCHEMBL2863210 0.87 CCR1 (0.50) P2RX7CCR1SMOMAPK1
SCHEMBL2852545 0.86 NPBWR1 (0.42) CCR1SMOALDH1A1MAPK1
SCHEMBL2853809 0.86 P2RX7 (0.49) P2RX7ALDH1A1
SCHEMBL2852356 0.85 CCR1 (0.48) P2RX7CCR1SMOMAPK1
SCHEMBL2855710 0.85 LMNA (0.46) P2RX7CCR1SMOMAPK1
SCHEMBL2854804 0.85 MAPK1 (0.48) P2RX7CCR1SMOALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed