SCHEMBL28525708

SCHEMBL28525708

O=[N+]([O-])c1ccc(N2CC(c3ccc(C(F)(F)F)cc3)C[C@@H]2CO)cc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 4/20 0.44
HTR1A P08908 1/20 0.40
TGM2 P21980 1/20 0.38
SLC6A9 P48067 1/20 0.36
SLC6A5 Q9Y345 1/20 0.36
SLC18A3 Q16572 1/20 0.35
HTR2C P28335 2/20 0.35
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ACHE P22303 1/20 0.34
GBA1 P04062 1/20 0.34
MMP1 P03956 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28531773 1.00 ENPP2 (0.44) ENPP2HTR1ATGM2SLC6A9SLC6A5
SCHEMBL28537640 0.90 ENPP2 (0.44) ENPP2HTR1ATGM2SLC6A9SLC6A5
SCHEMBL28547080 0.86 ENPP2 (0.40) ENPP2HTR1ATGM2MAPTACHE
SCHEMBL28542506 0.86 ENPP2 (0.40) ENPP2HTR1ATGM2MAPTACHE
SCHEMBL30474459 0.84 MAPT (0.39) ENPP2TGM2MAPTRAB9ANPSR1
SCHEMBL21616681 0.84 MAPT (0.39) ENPP2TGM2MAPTRAB9ANPSR1
SCHEMBL21616589 0.82 HTR2C (0.38) HTR2C
SCHEMBL21616638 0.82 HTR2C (0.38) HTR2C
SCHEMBL28529253 0.82 ENPP2 (0.42) ENPP2HTR1ATGM2SLC6A9SLC6A5
SCHEMBL28532309 0.82 ENPP2 (0.42) ENPP2HTR1ATGM2SLC6A9SLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed