SCHEMBL28532309

SCHEMBL28532309

O=C(O)[C@H]1CC(c2ccc(C(F)(F)F)cc2)CN1c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.42
HTR1A P08908 1/20 0.42
NOTUM Q6P988 1/20 0.39
SERPINE1 P05121 1/20 0.38
SLC6A9 P48067 1/20 0.38
SLC6A5 Q9Y345 1/20 0.38
TGM2 P21980 1/20 0.38
RAB9A P51151 2/20 0.37
PDE5A O76074 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ACHE P22303 1/20 0.36
POLB P06746 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PTPN1 P18031 1/20 0.36
PTPN6 P29350 1/20 0.36
PTPN11 Q06124 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28529253 1.00 ENPP2 (0.42) ENPP2HTR1ANOTUMSERPINE1SLC6A9
SCHEMBL28543121 0.87 MMP2 (0.45) ENPP2HTR1AMAPTPOLB
SCHEMBL28547111 0.87 MMP2 (0.45) ENPP2HTR1AMAPTPOLB
SCHEMBL28543125 0.87 MMP2 (0.45) ENPP2HTR1AMAPTPOLB
SCHEMBL28525708 0.82 ENPP2 (0.44) ENPP2HTR1ASLC6A9SLC6A5TGM2
SCHEMBL28531773 0.82 ENPP2 (0.44) ENPP2HTR1ASLC6A9SLC6A5TGM2
SCHEMBL28547080 0.78 ENPP2 (0.40) ENPP2HTR1ATGM2MAPTACHE
SCHEMBL28542506 0.78 ENPP2 (0.40) ENPP2HTR1ATGM2MAPTACHE
SCHEMBL13570060 0.77 ENPP2 (0.44) ENPP2HTR1ASLC6A9SLC6A5TGM2
SCHEMBL28537640 0.77 ENPP2 (0.44) ENPP2HTR1ASLC6A9SLC6A5TGM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed