SCHEMBL28537640

SCHEMBL28537640

O=[N+]([O-])c1ccc(N2CC(c3ccc(C(F)(F)F)cc3)CC[C@H]2CO)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 4/20 0.44
HTR1A P08908 1/20 0.39
TGM2 P21980 1/20 0.37
SLC18A3 Q16572 1/20 0.37
HTR2C P28335 2/20 0.36
SLC6A9 P48067 1/20 0.35
SLC6A5 Q9Y345 1/20 0.35
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28525708 0.90 ENPP2 (0.44) ENPP2HTR1ATGM2SLC18A3HTR2C
SCHEMBL28531773 0.90 ENPP2 (0.44) ENPP2HTR1ATGM2SLC18A3HTR2C
SCHEMBL28526930 0.85 HTR1A (0.39) ENPP2HTR1ATGM2ALDH1A1POLB
SCHEMBL23632290 0.82 SRD5A2 (0.43) HTR1A
SCHEMBL21616646 0.82 SRD5A2 (0.43) HTR1A
SCHEMBL21616615 0.80 HSD11B1 (0.42) HTR2C
SCHEMBL23632362 0.80 HSD11B1 (0.42) HTR2C
SCHEMBL23632570 0.79 ALDH1A1 (0.45) ALDH1A1POLBSMN1; SMN2
SCHEMBL28534482 0.79 ALDH1A1 (0.45) ALDH1A1POLBSMN1; SMN2
SCHEMBL28547080 0.79 ENPP2 (0.40) ENPP2HTR1ATGM2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed