SCHEMBL28525830

SCHEMBL28525830

CC(C)(C)OC(=O)N1CCC(c2cc(F)c3c(c2)NC(=O)CO3)C1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
PDE4B Q07343 1/20 0.43
HRH3 Q9Y5N1 4/20 0.39
GPR119 Q8TDV5 4/20 0.39
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
DPP4 P27487 1/20 0.39
TRPV3 Q8NET8 1/20 0.38
HPGDS O60760 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
IDH1 O75874 1/20 0.37
USP30 Q70CQ3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18305073 0.86 NR3C1 (0.39) MAPTPDE4BPOLB
SCHEMBL18305086 0.85 NR3C1 (0.37) MAPTPOLB
SCHEMBL28525837 0.84 MAPT (0.45) KDM4EMAPTTHRBPDE4BHRH3
SCHEMBL28907822 0.82 PDE4B (0.52) KDM4EMAPTTHRBPDE4BDDB1
SCHEMBL24582307 0.76 GPR119 (0.38) KDM4EMAPTTHRBGPR119DDB1
SCHEMBL28298497 0.75 PDE4B (0.56) KDM4EMAPTTHRBPDE4BGPR119
SCHEMBL28297779 0.75 PDE4B (0.56) KDM4EMAPTTHRBPDE4BGPR119
SCHEMBL30659460 0.73 DDB1 (0.47) KDM4EMAPTTHRBGPR119DDB1
SCHEMBL31565100 0.73 DDB1 (0.46) KDM4EMAPTTHRBGPR119DDB1
SCHEMBL26985427 0.72 PDE4B (0.58) KDM4EMAPTTHRBPDE4BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107873031-B Benzoxazinone derivatives and analogs thereof as modulators of TNF activity UCB生物制药私人有限公司 2021-03-12 CN disclosed