SCHEMBL28527136

SCHEMBL28527136

O=C(NCCN1CCOCC1)c1cn(-c2ccccc2)c2nc(NCc3ccccc3)ncc2c1=O

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 8/20 0.56
KDM5B Q9UGL1 6/20 0.48
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 2/20 0.46
HPGD P15428 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
HTT P42858 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28522950 0.95 CSF1R (0.53) CSF1RALDH1A1HPGDKDM4ELMNA
SCHEMBL28536148 0.89 CSF1R (0.58) CSF1RKDM5B
SCHEMBL3290842 0.87 CSF1R (0.62) CSF1RKDM5B
SCHEMBL3290621 0.85 CSF1R (0.75) CSF1R
SCHEMBL28527347 0.85 CSF1R (0.57) CSF1RALDH1A1HPGDKDM4E
SCHEMBL28528317 0.84 CSF1R (0.54) CSF1R
SCHEMBL3290854 0.84 CSF1R (0.56) CSF1RALDH1A1KMT2AKDM4EMEN1
SCHEMBL4796017 0.83 CSF1R (0.59) CSF1RALDH1A1KMT2AKDM4EMEN1
SCHEMBL28530641 0.83 CSF1R (0.62) CSF1RALDH1A1KMT2AMEN1
SCHEMBL3293656 0.82 CSF1R (0.69) CSF1RKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111848613-B Diaryl pyrimidopyridinone derivative and preparation method and application thereof 山东大学 2021-09-24 CN claimed
CN-111848613-A Diaryl pyrimidopyridinone derivative and preparation method and application thereof 山东大学 2020-10-30 CN claimed
CN-111848613-B Diaryl pyrimidopyridinone derivative and preparation method and application thereof 山东大学 2021-09-24 CN disclosed
CN-111848613-A Diaryl pyrimidopyridinone derivative and preparation method and application thereof 山东大学 2020-10-30 CN disclosed