SCHEMBL28528003

SCHEMBL28528003

COc1ccc(S(=O)(=O)OC(N)=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 3/20 0.56
PRSS1 P07477 3/20 0.56
PRSS2 P07478 3/20 0.56
PRSS3 P35030 3/20 0.56
PKM P14618 2/20 0.55
CA1 P00915 4/20 0.52
CA2 P00918 4/20 0.52
PARP10 Q53GL7 2/20 0.52
PARP1 P09874 1/20 0.52
PARP2 Q9UGN5 1/20 0.52
PARP4 Q9UKK3 1/20 0.52
GAA P10253 2/20 0.52
MMP1 P03956 1/20 0.52
MMP2 P08253 1/20 0.52
MMP9 P14780 1/20 0.52
MMP8 P22894 1/20 0.52
MMP13 P45452 1/20 0.52
CA9 Q16790 2/20 0.50
CA12 O43570 1/20 0.50
CA7 P43166 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27880969 0.85 PKM (0.55) F2PRSS1PRSS2PRSS3PKM
SCHEMBL8843455 0.82 F2 (0.50) F2PRSS1PRSS2PRSS3PKM
SCHEMBL28763397 0.80 F2 (0.53) F2PRSS1PRSS2PRSS3PKM
SCHEMBL28303054 0.80 ALDH1A1 (0.41) F2PRSS1PRSS2PRSS3PKM
SCHEMBL3836056 0.80 ALDH1A1 (0.58) F2PRSS1PRSS2PRSS3CA1
SCHEMBL8827511 0.78 TSHR (0.52) F2PRSS1PRSS2PRSS3PKM
SCHEMBL8198936 0.77 PKM (0.67) F2PRSS1PRSS2PRSS3PKM
SCHEMBL10763646 0.77 PKM (0.67) F2PRSS1PRSS2PRSS3PKM
SCHEMBL29221716 0.77 HSD11B1 (0.53) CA1CA2CA9ALDH1A1NPSR1
SCHEMBL18007730 0.76 F2 (0.50) F2PRSS1PRSS2PRSS3CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112367983-A 1,4 substituted isoquinoline inhibitors of KEAP1/NRF2 protein-protein interaction 伊利诺伊大学评议会 2021-02-12 CN disclosed