SCHEMBL2852839

SCHEMBL2852839

O=C(NCCc1ccc(O)c(O)c1)Oc1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.40
MAPT P10636 3/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
PTGS1 P23219 1/20 0.39
BLM P54132 1/20 0.39
HIF1A Q16665 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CCR1 P32246 3/20 0.38
TAAR1 Q96RJ0 1/20 0.38
ABCB1 P08183 1/20 0.38
P2RX7 Q99572 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
SPHK2 Q9NRA0 1/20 0.37
SPHK1 Q9NYA1 1/20 0.37
CETP P11597 1/20 0.37
PTPN7 P35236 1/20 0.37
DUSP3 P51452 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2860669 0.91 TAAR1 (0.46) MAPTKDM4EALDH1A1LMNACCR1
SCHEMBL2852955 0.91 KDM4E (0.44) SLC7A5MAPTKDM4EALDH1A1LMNA
SCHEMBL2853462 0.90 TRPV1 (0.42) MAPTCCR1TAAR1ABCB1P2RX7
SCHEMBL2850618 0.90 MAPT (0.44) MAPTLMNACCR1TAAR1ABCB1
SCHEMBL2857238 0.88 CCR1 (0.43) MAPTLMNACCR1TAAR1ABCB1
SCHEMBL2857600 0.88 CNR1 (0.46) MAPTCCR1TAAR1ABCB1P2RX7
SCHEMBL2852505 0.88 ABCB1 (0.48) MAPTALDH1A1LMNAHPGDHIF1A
SCHEMBL2860458 0.88 TP53 (0.46) MAPTLMNATAAR1P2RX7NPSR1
SCHEMBL2850857 0.88 TP53 (0.46) MAPTLMNATAAR1P2RX7NPSR1
SCHEMBL2854891 0.87 ABCB1 (0.52) ALDH1A1LMNAABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed