SCHEMBL2854891

SCHEMBL2854891

COc1ccc(CCNC(=O)Oc2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.52
GAA P10253 2/20 0.52
ALDH1A1 P00352 1/20 0.51
CNR1 P21554 1/20 0.50
LMNA P02545 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TP53 P04637 2/20 0.47
THRB P10828 1/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2857856 0.92 TSHR (0.49) ALDH1A1SMN1; SMN2CA12CA1CA2
SCHEMBL2850868 0.91 ALDH1A1 (0.51) ABCB1ALDH1A1SMN1; SMN2TP53CA12
SCHEMBL2860669 0.90 TAAR1 (0.46) ABCB1ALDH1A1CNR1LMNATP53
SCHEMBL2857600 0.88 CNR1 (0.46) ABCB1GAACNR1TP53
SCHEMBL2848475 0.88 CNR1 (0.48) ABCB1GAACNR1TP53
SCHEMBL2853462 0.88 TRPV1 (0.42) ABCB1CNR1
SCHEMBL2863131 0.88 CNR1 (0.50) ABCB1CNR1CA1CA2
SCHEMBL2852839 0.87 SLC7A5 (0.40) ABCB1ALDH1A1LMNA
SCHEMBL2852505 0.86 ABCB1 (0.48) ABCB1GAAALDH1A1CNR1LMNA
SCHEMBL2860458 0.86 TP53 (0.46) CNR1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed