SCHEMBL28528951

SCHEMBL28528951

O=C(O)Cn1cnc2c(ccn2C2CC2)c1=O

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.44
ADORA2B P29275 1/20 0.44
SMN1; SMN2 Q16637 4/20 0.40
NPC1 O15118 5/20 0.39
RAB9A P51151 5/20 0.39
TP53 P04637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 3/20 0.38
TSHR P16473 1/20 0.38
FSCN1 Q16658 2/20 0.38
PTGS2 P35354 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21643683 0.82 RAB9A (0.53) NPC1RAB9ATP53KDM4EALDH1A1
SCHEMBL28539473 0.76 KDM4E (0.41) HDAC6ADORA2BSMN1; SMN2NPC1RAB9A
SCHEMBL13799935 0.69 SMN1; SMN2 (0.76) HDAC6SMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL21643688 0.69 POLB (0.40) TP53LMNA
SCHEMBL12878629 0.69 NPC1 (0.50) ADORA2BSMN1; SMN2NPC1RAB9ATP53
SCHEMBL28709455 0.68 TRPA1 (0.56) HDAC6SMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL20971253 0.66 ALDH1A1 (0.41) SMN1; SMN2ALDH1A1LMNAHTT
SCHEMBL17163964 0.66 TRPA1 (0.58) HDAC6ADORA2BSMN1; SMN2NPC1RAB9A
SCHEMBL23103466 0.65 GRM1 (0.38)
SCHEMBL10085099 0.65 HDAC6 (0.61) HDAC6SMN1; SMN2NPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513047-B Heteroaromatic NMDA receptor modulators and uses thereof 诺华股份有限公司 2023-10-20 CN disclosed
CN-112513047-A Heteroaromatic NMDA receptor modulators and uses thereof 卡登特治疗公司 2021-03-16 CN disclosed