SCHEMBL28529154

SCHEMBL28529154

COc1cccc(-c2cc(B(O)O)cs2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.56
HSD17B1 P14061 3/20 0.51
HSD17B2 P37059 3/20 0.51
HDAC6 Q9UBN7 1/20 0.44
ALDH1A1 P00352 4/20 0.42
MAPT P10636 3/20 0.42
HSD17B10 Q99714 2/20 0.42
LMNA P02545 2/20 0.42
ATP4A P20648 1/20 0.42
ATP4B P51164 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
DYRK1A Q13627 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
HPGD P15428 2/20 0.41
NPC1 O15118 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
IKBKB O14920 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28520492 0.80 MGLL (0.53) ENPP2HSD17B1HSD17B2ALDH1A1DYRK1A
SCHEMBL28528851 0.80 HSD17B1 (0.41) HSD17B1HSD17B2ALDH1A1MAPTHSD17B10
SCHEMBL1180286 0.79 HSD17B1 (0.56) HSD17B1HSD17B2HDAC6ALDH1A1MAPT
SCHEMBL1180161 0.78 HSD17B1 (0.52) HSD17B1HSD17B2HDAC6ALDH1A1MAPT
SCHEMBL28060965 0.77 ENPP2 (0.85) ENPP2HSD17B2HDAC4HDAC8DYRK1A
SCHEMBL28574792 0.76 HSD17B1 (0.51) HSD17B1HSD17B2HDAC6ALDH1A1MAPT
SCHEMBL20262887 0.76 ENPP2 (0.65) ENPP2HDAC4HDAC8DYRK1ACLK4
SCHEMBL1181055 0.75 ABL1 (0.53) HSD17B1HSD17B2HDAC6ALDH1A1HDAC4
SCHEMBL29742784 0.75 HSD17B1 (0.67) HSD17B1HSD17B2HDAC6ALDH1A1MAPT
SCHEMBL28635415 0.75 HSD17B1 (0.67) HSD17B1HSD17B2HDAC6ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602834-B Bruton's tyrosine kinase inhibitor 北京盛诺基医药科技股份有限公司 2021-01-08 CN disclosed