SCHEMBL28574792

SCHEMBL28574792

COc1cccc(-c2cc(Cl)cs2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.51
HSD17B2 P37059 1/20 0.51
LMNA P02545 2/20 0.47
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CNR1 P21554 2/20 0.45
DYRK1A Q13627 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
ALDH1A1 P00352 2/20 0.44
CYP19A1 P11511 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CYP1A1 P04798 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C8 P10632 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2A6 P11509 1/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1180286 0.83 HSD17B1 (0.56) HSD17B1HSD17B2LMNAMAPTKDM4E
SCHEMBL1180161 0.81 HSD17B1 (0.52) HSD17B1HSD17B2LMNAMAPTKDM4E
SCHEMBL1181055 0.79 ABL1 (0.53) HSD17B1HSD17B2DYRK1ACLK4ALDH1A1
SCHEMBL4947340 0.78 CNR1 (0.50) HSD17B1HSD17B2LMNAMAPTKDM4E
SCHEMBL23452051 0.78 HSD17B1 (0.49) HSD17B1HSD17B2LMNAMAPTKDM4E
SCHEMBL1180026 0.77 ABL1 (0.54) HSD17B1HSD17B2DYRK1ACLK4ALDH1A1
SCHEMBL28529154 0.76 ENPP2 (0.56) HSD17B1HSD17B2LMNAMAPTKDM4E
SCHEMBL29742784 0.75 HSD17B1 (0.67) HSD17B1HSD17B2LMNAMAPTALDH1A1
SCHEMBL28635415 0.75 HSD17B1 (0.67) HSD17B1HSD17B2LMNAMAPTALDH1A1
SCHEMBL12093643 0.75 HDAC6 (0.55) HSD17B1HSD17B2MAPTTDP1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218878-A NTCP inhibitors 北京生命科学研究所 2021-01-12 CN disclosed