SCHEMBL28529935

SCHEMBL28529935

C=C[C@@]1(COCc2ccccc2)CC[C@@H](c2cccc(F)c2)N1C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.40
RIPK1 Q13546 2/20 0.39
TACR1 P25103 1/20 0.39
GPR119 Q8TDV5 1/20 0.37
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
PDE5A O76074 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
NR1H2 P55055 3/20 0.34
RXRA P19793 2/20 0.34
NR1H3 Q13133 2/20 0.34
TP53 P04637 1/20 0.34
BACE1 P56817 1/20 0.34
BACE2 Q9Y5Z0 1/20 0.34
USP30 Q70CQ3 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28907234 0.92 PKM (0.41) PKMRIPK1TACR1GPR119ALDH1A1
SCHEMBL20835550 0.90 PKM (0.42) PKMRIPK1ALDH1A1LMNAMAOA
SCHEMBL28515213 0.84 PKM (0.41) PKMRIPK1TACR1GPR119ALDH1A1
SCHEMBL20835738 0.82 PKM (0.43) PKMRIPK1ALDH1A1LMNAMAOA
SCHEMBL20835589 0.81 PKM (0.43) PKMRIPK1TACR1GPR119ALDH1A1
SCHEMBL28529951 0.80 RIPK1 (0.44) RIPK1GPR119ALDH1A1PDE5AMAOB
SCHEMBL28518960 0.79 RIPK1 (0.40) PKMRIPK1GPR119NR1H2RXRA
SCHEMBL31479820 0.76 RIPK1 (0.47) PKMRIPK1GPR119ALDH1A1PDE5A
SCHEMBL20835834 0.74 PKM (0.43) PKMRIPK1ALDH1A1LMNAMEN1
SCHEMBL28515805 0.73 CALCRL (0.47) RIPK1GPR119ALDH1A1PDE5APSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109476639-B Pyrrolidine derivatives 橘生药品工业股份有限公司 2021-02-26 CN disclosed