SCHEMBL8209503

SCHEMBL8209503

NC(=O)c1cnn(Cc2ccc(C(F)(F)F)nc2)c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 5/20 0.45
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HSD17B10 Q99714 1/20 0.40
PPARD Q03181 1/20 0.40
LMNA P02545 2/20 0.40
GRM2 Q14416 4/20 0.39
KCNH2 Q12809 1/20 0.39
GPR119 Q8TDV5 1/20 0.39
MAPT P10636 1/20 0.39
NR1H2 P55055 1/20 0.37
S1PR1 P21453 1/20 0.37
S1PR3 Q99500 1/20 0.37
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30744539 0.87 PPARD (0.42) KLKB1KDM4EALDH1A1HSD17B10PPARD
SCHEMBL21493002 0.87 PPARD (0.42) KLKB1KDM4EALDH1A1HSD17B10PPARD
SCHEMBL27286166 0.83 KDM4E (0.49) KLKB1KDM4EALDH1A1HSD17B10LMNA
SCHEMBL17685622 0.82 KLKB1 (0.46) KLKB1KDM4EALDH1A1HSD17B10LMNA
SCHEMBL28532124 0.81 PPARD (0.39) KLKB1KDM4EALDH1A1HSD17B10PPARD
SCHEMBL21491889 0.79 KLKB1 (0.44) KLKB1PPARD
SCHEMBL21503682 0.79 LOXL2 (0.40) KLKB1PPARDLMNAKCNH2MAPT
Hydrochloric Acid SCHEMBL21491894 0.77 LMNA (0.41) KLKB1PPARDLMNAKCNH2MAPT
Hydrochloric Acid SCHEMBL30744436 0.77 LMNA (0.41) KLKB1PPARDLMNAKCNH2MAPT
SCHEMBL25269987 0.77 GRIN1 (0.40) PPARDLMNAKCNH2GPR119MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188099-B2 Method of decreasing hepatotoxic side effects using A2B adenosine receptor antagonists GILEAD SCIENCES, INC. (US) 2012-05-29 US disclosed