SCHEMBL28533641

SCHEMBL28533641

C[C@H]1Oc2c(F)cc(-c3ccn(C(=O)OC(C)(C)C)c3)cc2NC1=O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 4/20 0.35
BRD4 O60885 4/20 0.35
LIPC P11150 1/20 0.32
LIPG Q9Y5X9 1/20 0.32
PARP1 P09874 7/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
CECR2 Q9BXF3 1/20 0.31
DRD2 P14416 2/20 0.31
RXRA P19793 3/20 0.30
NR1H2 P55055 3/20 0.30
NR1H3 Q13133 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20138131 0.86 PARP1 (0.34) CREBBPBRD4PARP1PDE3BPDE3A
SCHEMBL28909618 0.81 NR3C2 (0.43) CREBBPBRD4LIPCLIPGDRD2
SCHEMBL28525837 0.71 MAPT (0.45)
SCHEMBL18128118 0.68 PARP1 (0.38) BRD4PARP1PDE3BPDE3ADRD2
SCHEMBL18127979 0.68 PARP1 (0.38) BRD4PARP1PDE3BPDE3ADRD2
SCHEMBL28907820 0.67 KDM4E (0.45) PARP1PDE3BPDE3A
SCHEMBL20137948 0.67 CYP11B2 (0.41) PARP1PDE3BPDE3A
SCHEMBL18128043 0.67 PARP1 (0.44) BRD4PARP1PDE3BPDE3ACECR2
SCHEMBL30806796 0.67 PARP1 (0.44) BRD4PARP1PDE3BPDE3ACECR2
SCHEMBL16792483 0.67 PARP1 (0.44) BRD4PARP1PDE3BPDE3ACECR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107873031-B Benzoxazinone derivatives and analogs thereof as modulators of TNF activity UCB生物制药私人有限公司 2021-03-12 CN disclosed