SCHEMBL28536397

SCHEMBL28536397

O=C(/C=C/c1ccc(F)cc1)Oc1ccc(F)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.62
KMT2A Q03164 6/20 0.62
MEN1 O00255 3/20 0.59
TNFRSF1A P19438 1/20 0.56
KDM4E B2RXH2 1/20 0.56
GAA P10253 1/20 0.56
POLB P06746 1/20 0.54
MAPT P10636 1/20 0.53
MAOB P27338 1/20 0.53
LMNA P02545 1/20 0.50
CTSL P07711 1/20 0.50
NFE2L2 Q16236 1/20 0.50
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBA3C P0DPH7 1/20 0.50
TUBA1B P68363 1/20 0.50
TUBA4A P68366 1/20 0.50
TUBB4B P68371 1/20 0.50
TUBB3 Q13509 1/20 0.50
TUBB2A Q13885 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28545557 0.93 CA12 (0.57) HSD11B1KMT2AMEN1TNFRSF1AKDM4E
SCHEMBL28542113 0.92 KMT2A (0.57) HSD11B1KMT2AMEN1TNFRSF1AKDM4E
SCHEMBL27737751 0.92 KMT2A (0.54) HSD11B1KMT2AMEN1TNFRSF1AKDM4E
SCHEMBL28541241 0.89 CYP2D6 (0.52) HSD11B1KMT2AMEN1TNFRSF1AKDM4E
SCHEMBL27758520 0.86 MAOB (0.66) KMT2AMEN1MAPTMAOBLMNA
SCHEMBL28894377 0.86 KMT2A (0.48) HSD11B1KMT2AMEN1TNFRSF1AKDM4E
SCHEMBL11215369 0.85 MAOB (0.58) KMT2AMEN1KDM4EGAAPOLB
SCHEMBL11215372 0.85 MAOB (0.58) KMT2AMEN1KDM4EGAAPOLB
SCHEMBL21848007 0.84 HSD11B1 (0.67) HSD11B1KMT2AMEN1TNFRSF1APOLB
SCHEMBL776127 0.84 HSD11B1 (0.67) HSD11B1KMT2AMEN1TNFRSF1APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112624927-B TRPV3 inhibitor and preparation method thereof 青岛大学 2023-07-21 CN disclosed
CN-112691099-B Application of organic compound in preparation of medicine for treating colon cancer 青岛大学 2022-09-30 CN disclosed
CN-112691099-A Application of organic compound in preparation of medicine for treating colon cancer 青岛大学 2021-04-23 CN disclosed
CN-112624927-A TRPV3 inhibitor and preparation method thereof 青岛大学 2021-04-09 CN disclosed