SCHEMBL28545557

SCHEMBL28545557

O=C(/C=C/c1ccc(O)cc1)Oc1ccc(F)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.57
CA1 P00915 4/20 0.57
CA2 P00918 4/20 0.57
CA7 P43166 4/20 0.57
CA9 Q16790 4/20 0.57
CA14 Q9ULX7 4/20 0.57
TYR P14679 3/20 0.57
MMP1 P03956 1/20 0.56
MMP2 P08253 1/20 0.56
MMP9 P14780 1/20 0.56
KMT2A Q03164 4/20 0.55
MEN1 O00255 3/20 0.55
MAPT P10636 1/20 0.55
HSD11B1 P28845 2/20 0.55
AKR1B10 O60218 2/20 0.53
AKR1B1 P15121 2/20 0.53
CTSL P07711 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
F3 P13726 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28536397 0.93 HSD11B1 (0.62) KMT2AMEN1MAPTHSD11B1CTSL
SCHEMBL29009143 0.91 CA12 (0.67) CA12CA1CA2CA7CA9
SCHEMBL27737751 0.85 KMT2A (0.54) KMT2AMEN1MAPTHSD11B1CTSL
SCHEMBL28542113 0.85 KMT2A (0.57) KMT2AMEN1MAPTHSD11B1CTSL
SCHEMBL149407 0.85 CA12 (0.72) CA12CA1CA2CA7CA9
SCHEMBL5966380 0.85 CA12 (0.72) CA12CA1CA2CA7CA9
SCHEMBL679710 0.85 CA12 (0.72) CA12CA1CA2CA7CA9
SCHEMBL14877836 0.83 MAPT (0.77) CA12CA1CA2CA7CA9
SCHEMBL20102637 0.83 ESR1 (0.61) CA12CA1CA2CA7CA9
SCHEMBL22005455 0.83 MAPT (0.77) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112624927-B TRPV3 inhibitor and preparation method thereof 青岛大学 2023-07-21 CN disclosed
CN-112691099-B Application of organic compound in preparation of medicine for treating colon cancer 青岛大学 2022-09-30 CN disclosed
CN-112691099-A Application of organic compound in preparation of medicine for treating colon cancer 青岛大学 2021-04-23 CN disclosed
CN-112624927-A TRPV3 inhibitor and preparation method thereof 青岛大学 2021-04-09 CN disclosed