SCHEMBL28538296

SCHEMBL28538296

Fc1cc(N2CCCC2c2ccccc2C2CC2)ccc1Br

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
TSHR P16473 2/20 0.36
AR P10275 1/20 0.34
MAPT P10636 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRK1 P41145 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28528284 0.81 CYP2D6 (0.38) KMT2ACYP2C9CYP2C19TSHROPRM1
SCHEMBL28528279 0.81 CYP2D6 (0.38) KMT2ACYP2C9CYP2C19TSHROPRM1
SCHEMBL28534879 0.80 OPRM1 (0.39) ALDH1A1KMT2AOPRM1OPRK1
SCHEMBL28519576 0.77 NOS1 (0.37) ALDH1A1GAAKMT2AMAPTOPRM1
SCHEMBL24775580 0.77 HRH3 (0.38) CYP2C9CYP2C19MAPTOPRM1OPRK1
SCHEMBL28535286 0.75 CHRNB2 (0.40) OPRM1OPRK1
SCHEMBL31525091 0.73 HTR2C (0.41) CYP2C9CYP2C19
SCHEMBL28909558 0.73 HRH3 (0.41) CYP2C9CYP2C19MAPTOPRM1OPRK1
SCHEMBL28909552 0.73 HRH3 (0.41) CYP2C9CYP2C19MAPTOPRM1OPRK1
SCHEMBL28529792 0.73 HTR2C (0.41) CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117683029-A Bcl-2 inhibitors 百济神州有限公司 2024-03-12 CN disclosed
CN-117430601-A Bcl-2 inhibitors 百济神州有限公司 2024-01-23 CN disclosed
CN-112437772-B Bcl-2 inhibitors 百济神州有限公司 2023-11-21 CN disclosed
CN-112437772-A Bcl-2 inhibitors 百济神州有限公司 2021-03-02 CN disclosed