SCHEMBL28544472

SCHEMBL28544472

CC(=O)Nc1cc(F)c([N+](=O)[O-])cc1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.52
NPSR1 Q6W5P4 2/20 0.52
ALDH1A1 P00352 2/20 0.52
LMNA P02545 2/20 0.52
GALR2 O43603 1/20 0.52
MITF O75030 1/20 0.52
POLB P06746 1/20 0.52
HSP90AA1 P07900 1/20 0.52
HPGD P15428 1/20 0.52
XBP1 P17861 1/20 0.52
CCR6 P51684 1/20 0.52
AKR1C2 P52895 3/20 0.48
AKR1C1 Q04828 1/20 0.48
MAPT P10636 3/20 0.46
GAA P10253 1/20 0.45
SLC9A1 P19634 1/20 0.45
KDM4E B2RXH2 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HTT P42858 3/20 0.43
AKR1C3 P42330 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5167381 0.94 SMN1; SMN2 (0.52) SMN1; SMN2NPSR1ALDH1A1LMNAGALR2
SCHEMBL1965597 0.88 NPSR1 (0.49) SMN1; SMN2NPSR1ALDH1A1LMNAGALR2
SCHEMBL14854666 0.86 ALDH1A1 (0.60) SMN1; SMN2NPSR1ALDH1A1LMNAGALR2
SCHEMBL671475 0.85 MAPT (0.55) SMN1; SMN2LMNAAKR1C2AKR1C1MAPT
SCHEMBL4652737 0.84 MAPT (0.54) SMN1; SMN2NPSR1ALDH1A1LMNAGALR2
SCHEMBL3251790 0.84 NPSR1 (0.50) SMN1; SMN2NPSR1ALDH1A1LMNAGALR2
SCHEMBL30748250 0.84 NPSR1 (0.50) SMN1; SMN2NPSR1ALDH1A1LMNAGALR2
SCHEMBL23070353 0.84 SMN1; SMN2 (0.57) SMN1; SMN2NPSR1ALDH1A1LMNAGALR2
SCHEMBL7375343 0.82 SLC9A1 (0.61) SMN1; SMN2NPSR1ALDH1A1LMNAGALR2
SCHEMBL4149265 0.82 LMNA (0.48) SMN1; SMN2NPSR1ALDH1A1LMNAGALR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112707845-B Preparation method of dacatinib intermediate 成都伊诺达博医药科技有限公司 2023-04-28 CN disclosed
CN-112707845-A Preparation method of dacomitinib intermediate 成都伊诺达博医药科技有限公司 2021-04-27 CN disclosed