SCHEMBL28545378

SCHEMBL28545378

CCOC(=O)c1ccc(Nc2ccc(F)c(F)c2)cn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
DHODH Q02127 4/20 0.46
TTK P33981 1/20 0.46
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
KDM4E B2RXH2 2/20 0.45
P2RY12 Q9H244 1/20 0.45
LMNA P02545 3/20 0.43
KCNQ3 O43525 1/20 0.42
KCNQ2 O43526 1/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 1/20 0.42
CASP3 P42574 1/20 0.42
KMT2A Q03164 1/20 0.42
TRPV1 Q8NER1 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
ALDH1A1 P00352 1/20 0.42
SYK P43405 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28532069 0.87 ALDH1A1 (0.54) SMN1; SMN2NPC1RAB9AHPGDKDM4E
SCHEMBL28545895 0.86 MAPT (0.46) SMN1; SMN2RAB9ATSHRKDM4ELMNA
SCHEMBL28532052 0.85 HTT (0.56) SMN1; SMN2NPC1RAB9AHPGDKDM4E
SCHEMBL29031128 0.82 SMN1; SMN2 (0.47) SMN1; SMN2NPC1RAB9AHPGDKDM4E
SCHEMBL29031101 0.82 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9AHPGDKDM4E
SCHEMBL28543158 0.81 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9ADHODHHPGD
SCHEMBL28537077 0.81 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9ATSHRKDM4E
SCHEMBL28540429 0.80 MTNR1B (0.62) SMN1; SMN2NPC1RAB9AHPGDKDM4E
SCHEMBL28545384 0.79 CYP1A2 (0.43) SMN1; SMN2NPC1RAB9ADHODHTSHR
SCHEMBL28543171 0.79 PDE4B (0.51) SMN1; SMN2NPC1RAB9ADHODHKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111925357-B Acylhydrazone compound, pharmaceutical composition and application thereof 中国科学院昆明植物研究所 2023-06-06 CN disclosed
CN-111925357-A Acylhydrazone compound, pharmaceutical composition and application thereof 中国科学院昆明植物研究所 2020-11-13 CN disclosed