SCHEMBL28545686

SCHEMBL28545686

CC(=O)Nc1ccc(Cl)c(C)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 1/20 0.51
SCN9A Q15858 1/20 0.48
SCN2A Q99250 1/20 0.48
SCN3A Q9NY46 1/20 0.48
SCN10A Q9Y5Y9 1/20 0.48
SORT1 Q99523 1/20 0.47
KDM4E B2RXH2 3/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
ADORA3 P0DMS8 3/20 0.43
DYRK1A Q13627 1/20 0.43
FSCN1 Q16658 1/20 0.43
MAPK8 P45983 1/20 0.41
ABL1 P00519 2/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753194 0.81 SORT1 (0.53) PTK2SORT1KDM4ELMNAL3MBTL1
SCHEMBL27342111 0.81 SCN10A (0.51) SCN10ASORT1KDM4EMAPTL3MBTL1
SCHEMBL21723677 0.81 ALDH1A1 (0.51) SORT1KDM4ELMNAMAPTNPC1
SCHEMBL28552164 0.80 RAB9A (0.45) SORT1LMNAMAPTL3MBTL1NPC1
SCHEMBL1269767 0.78 RAB9A (0.60) KDM4ELMNAMAPTL3MBTL1NPC1
SCHEMBL27398574 0.78 PTK2 (0.51) PTK2SCN9ASCN2ASCN3ASCN10A
SCHEMBL2019170 0.78 KDM4E (0.46) PTK2SCN9ASCN2ASCN3ASCN10A
SCHEMBL7092192 0.78 SMN1; SMN2 (0.48) PTK2SORT1KDM4ELMNAMAPT
SCHEMBL19736135 0.78 GRM5 (0.50) PTK2SCN9ASCN2ASCN3ASCN10A
SCHEMBL9974219 0.78 KDM4E (0.46) PTK2SCN9ASCN2ASCN3ASCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112654354-A 1,3,4, 9-tetrahydro-2H-pyrido [3,4-b ] indole derivative compound and application thereof 菲尼克思药业股份有限公司 2021-04-13 CN disclosed