SCHEMBL2854586

SCHEMBL2854586

COc1cccc(CCNC(=O)Oc2cnn(-c3ccccc3)c2C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
HTT P42858 1/20 0.47
GAA P10253 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
DGAT2 Q96PD7 1/20 0.46
KDM4E B2RXH2 3/20 0.46
TOP2A P11388 1/20 0.45
TSHR P16473 1/20 0.45
SPR P35270 1/20 0.44
LMNA P02545 1/20 0.43
MAPT P10636 2/20 0.43
POLB P06746 2/20 0.43
IDO1 P14902 1/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852556 0.93 TDP1 (0.44) ALDH1A1MEN1KMT2ANPSR1GAA
SCHEMBL2859429 0.93 NPC1 (0.46) ALDH1A1MEN1KMT2ASMN1; SMN2NPSR1
SCHEMBL2863131 0.92 CNR1 (0.50) MEN1KMT2ANPSR1HTTTAAR1
SCHEMBL2852633 0.90 TAAR1 (0.57) ALDH1A1MEN1KMT2AGAANPC1
SCHEMBL2854509 0.88 KDM4E (0.50) ALDH1A1SMN1; SMN2GAANPC1RAB9A
SCHEMBL2850868 0.88 ALDH1A1 (0.51) ALDH1A1KMT2ASMN1; SMN2HTTMAPT
SCHEMBL2857230 0.88 KDM4E (0.44) ALDH1A1SMN1; SMN2NPSR1HTTGAA
SCHEMBL2863198 0.88 CCR1 (0.50) ALDH1A1SMN1; SMN2NPSR1KDM4EMAPT
SCHEMBL2853061 0.88 KDM4E (0.44) ALDH1A1SMN1; SMN2NPC1RAB9ATAAR1
SCHEMBL2852221 0.87 ALDH1A1 (0.46) ALDH1A1MEN1KMT2ASMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed