SCHEMBL2854730

SCHEMBL2854730

Cc1ccccc1C(=O)C#CC(=O)NC1CCN(c2nc(C(C)(C)C)cs2)C1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
KCNH2 Q12809 1/20 0.37
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
PAK1 Q13153 1/20 0.36
ACKR3 P25106 3/20 0.35
PDE10A Q9Y233 2/20 0.35
BTK Q06187 4/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
POLB P06746 2/20 0.34
ALOX15 P16050 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
CCR4 P51679 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855060 0.91 ALDH1A1 (0.43) ALDH1A1PAK1ACKR3BTKMEN1
SCHEMBL973611 0.86 LMNA (0.37) CTSBCTSSCTSKKCNH2LMNA
SCHEMBL2853786 0.86 LMNA (0.38) CTSBCTSSCTSKKCNH2ALDH1A1
SCHEMBL2858190 0.84 MEN1 (0.38) CTSBCTSSCTSKKCNH2ALDH1A1
SCHEMBL974388 0.83 DRD2 (0.43) CTSBCTSSCTSKKCNH2ALDH1A1
SCHEMBL2861257 0.83 SMN1; SMN2 (0.37) ALDH1A1PAK1ACKR3BTKMEN1
SCHEMBL972936 0.81 LMNA (0.39) CTSBCTSSCTSKKCNH2ALDH1A1
SCHEMBL974674 0.80 BTK (0.39) CTSBCTSSCTSKKCNH2LMNA
SCHEMBL973921 0.80 SMN1; SMN2 (0.38) CTSBCTSSCTSKKCNH2ALDH1A1
SCHEMBL973133 0.80 LMNA (0.38) CTSBCTSSCTSKKCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968957-B1 SUBSTITUTED THIAZOLES AND THEIR USE FOR PRODUCING DRUGS GRUENENTHAL GMBH (DE) 2010-01-20 EP claimed